The evolving small-molecule fluorescent-conjugate toolbox for Class A GPCRs
Structural and functional insights into the juxtamembranous amino-terminal tail and extracellular loop regions of class B GPCRs
Allosteric interactions at adenosine A1 and A3 receptors: new insights into the role of small molecules and receptor dimerization
Molecular mechanisms underlying physiological and receptor pleiotropic effects mediated by GLP-1R activation
The GPCR, class C, group 6, subtype A (GPRC6A) receptor: from cloning to physiological function
Engendering biased signalling from the calcium-sensing receptor for the pharmacotherapy of diverse disorders
GPBA: a GPCR for bile acids and an emerging therapeutic target for disorders of digestion and sensation
The structural role of receptor tyrosine sulfation in chemokine recognition
Biased signalling and proteinase-activated receptors (PARs): targeting inflammatory disease
WNT/Frizzled signalling: receptor–ligand selectivity with focus on FZD-G protein signalling and its physiological relevance: IUPHAR Review 3
Cell-specific blood–brain barrier regulation in health and disease: a focus on hypoxia
Should pharmacologists care about alternative splicing? IUPHAR Review 4
Unexpectedly high affinity of a novel histamine H3 receptor antagonist, GSK239512, in vivo in human brain, determined using PET
The ryanodine receptor agonist 4-chloro-3-ethylphenol blocks ORAI store-operated channels
TLR9 and MyD88 are crucial for the maturation and activation of dendritic cells by paromomycin–miltefosine combination therapy in visceral leishmaniasis
Hypotensive effects of ghrelin receptor agonists mediated through a novel receptor
The MCH1 receptor, an anti-obesity target, is allosterically inhibited by 8-methylquinoline derivatives possessing subnanomolar binding and long residence times
Deletion of thioredoxin-interacting protein preserves retinal neuronal function by preventing inflammation and vascular injury
Role of the A2B receptor–adenosine deaminase complex in colonic dysmotility associated with bowel inflammation in rats
Heterologous regulation of agonist-independent μ-opioid receptor phosphorylation by protein kinase C